Sr.No Chemical Name Therapeutic Category End Use CAS No
1 N-(2-Methyl-5-nitrophenyl)-4-(3-pyridyl)-2-pyrimidine Amine Antineoplastic Imatinib mesylate 152460-09-8
2 N-(5-Amino-2-Methylphenyl)-4-(3-pyridyl)-2-pyrimidineamine Antineoplastic Imatinib mesylate 152460-10-1
3 4-(4-Methyl piperazine-1-yl)methyl benzoic acid di HCl Antineoplastic Imatinib mesylate 106261-49-8
4 4-(4-Methyl piperazine-1-yl)methyl benzoyl chloride di HCl Antineoplastic Imatinib mesylate 106261-64-7
5 2-[3-(Cyano-Dimethyl-methyl)-5-methyl-phenyl]-2-methyl propionitrile Antineoplastic Anastrozole 120511-72-0
6 1,2,3,9-Tetrahydro-9-methyl-4(H)-Carbazol-4-One Antiemetic Ondansetron 27387-31-1
7 3-[(Dimethylamino)methyl]-1,2,3,9-tetrahydro-9-methyl-4H- carbazol-4-one HCl Antiemetic Ondansetron 119812-29-2
8 2-Amino-5-Methylthiophene-3-carbonitrile Antipsychotic Olanzapine 138564-58-6
9 2-(2-Aminophenylamino)-5-Methylthiophene-3-Carbonitrile Antipsychotic Olanzapine 873895-41-1
10 2-(2-Nitroanilino)-5-methylthiophene-3-carbonitrile (Grade-1) &  (Grade-2) Antipsychotic Olanzapine 138564-59-7
11 4-Amino-2-methyl-10H-thieno-[2,3-b][1,5]-benzodiazepine hydrochloride Antipsychotic Olanzapine 138564-60-0
12 (+/-)-1-Phenyl-1,2,3,4-Tetrahydro Isoquinoline  Renal and genitourinary agent Solifenacin Succinate 22990-19-8
13 (S)-1-Phenyl-1,2,3,4-Tetrahydro Isoquinoline (Grade-1) & (Grade-2)  Renal and genitourinary agent Solifenacin Succinate 118864-75-8
14 N-Formyl IsoNipecotic Acid atypical antipsychotic Risperidone
Paliperidone
Iloperidone
84163-42-8
15 2,4-Difluoro phenyl (4-Piperidinyl)Methanone Oxime HCl atypical antipsychotic Risperidone
Paliperidone
Iloperidone
135634-18-3
16 6-Fluoro-3-(4-piperadinyl)-1,2-benzisoxazole atypical antipsychotic Risperidone
Paliperidone
Iloperidone
84163-77-9
17 4-(6-Fluoro-1,2-benzisoxazole-3yl)-piperidine HCl (Grade-2) atypical antipsychotic Risperidone 84163-13-3
18 3-(N-Methyl-N-Pentyl amino)propionic acid HCl Bone Resorption Inhibitors Ibandronate sodium 625120-81-2
19 (1-Hydroxy-2-(3-pyridinyl)ethylidine)-1,1-bisphosphonic acid Calcium regulator Risedronate sodium 105462-24-6
20 R-9-(2-Hydroxy Propyl)adenine Antiretroviral Agent Tenofovir 14047-28-0
21 Imidazole-1yl-acetic acid Hydrochloride  Calcium Regulator. Zoledronic Acid 87266-37-3
22 Benzyl glycinate p-toluene sulfonate antidiarrheal Racecadotril 1738-76-7
23 9-(Benzyloxy)-3-(2-Chloroethyl)-2-Methyl-4H-Pyrido[1,2-A] Pyrimidin-4-one atypical antipsychotic Paliperidone 147687-17-0
24 3-(2-chloroethyl)-9-hydroxy-2-methyl-6,7,8,9-tetrahydropyrido[1,2-a] pyrimidin-4-one atypical antipsychotic Paliperidone 130049-82-0
25 1-(3-chloro propyl)-1,3-dihydro-2H-benzimidazol-2-one Antihistamine Oxatomide 62780-89-6
26 2,2-(5-bromo methyl-1,3-phenylene)di(2-methyl propionitrile) Antineoplastic Anastrozole 120511-84-4
27 9-[(R)-2-(Phosphonomethoxy) Propyl] adenine Monohydrate Antiretroviral Agent Tenofovir 206184-49-8
28 N-(4-methylAminobenzoyl)-L-glutamic acid diethyl ester Antineoplastic Methotrexate 2378-95-2
29 1-(4-(3-chloropropoxy)-3-methoxy phenyl)ethanone Antipsychotic Iloperidone 58113-30-7
30 (R)-(-)-3-Quinuclidinol hydrochloride  Renal and genitourinary agent Solifenacin succinate 42437-96-7
31 (S)-ethyl 1-phenyl-3,4-dihydroisoquinoline-2(1H)-carboxylate 180468-42-2
32 (R)-(-)-3-Quinuclidinol 25333-42-0
33 2-[(6-Chloro-3,4-dihydro-3-methyl-2,4-dioxo-1(2H)-pyrimidinyl)methyl]-Benzonitrile Anti Diabetic Alogliptin 865758-96-9
34 1-(4-Iodophenyl)-3-morpholino-5,6- dihydropyridin-2(III)-one Anti Coagulant Apixaban 473927-69-4
35 Chloro[(4-methoxy phenyl)hydrazono] acetic acid ethyl ester Anti Coagulant Apixaban 27143-07-3
36 4,5,6,7-tetrahydro-1-(4-methoxyphenyl)-7- oxo-6-(4-(2-oxopiperidin-1-yl)phenyl)-1H-pyrazolo [3,4-c]pyridine-3-carboxylic acid ethyl ester Anti Coagulant Apixaban 503614-91-3
37 2-Piperidone Anti Coagulant Apixaban 675-20-7
38 3-Morpholino-1-(4-(2-oxopiperidin-1-yl)-5,6-dihydropyridin-2(1H)-one Anti Coagulant Apixaban 545445-44-1
39 3-chloro-5,6-dihydropyridine-2(H)-one Anti Coagulant Apixaban
40 Ethyl 6-(4-iodophenyl)_1-(4-methoxyphenyl) 7-oxo-4,5,6,7-tetrahydro-1H-pyrazolo[3,4-c]pyridine-3-carboxylate Anti Coagulant Apixaban 473927-64-9
41 2,3,4,6-tetrakis-O-(trimethylsilyl)D-glocono 1,5-lactone Anti Diabetic Canagliflozin 32384-65-9
42 2-(5-bromo-2-methyl benzyl)-5-(4-fluorophenyl) thiophene Anti Diabetic Canagliflozin
43 (2R,3R,4S,5S,6R)-2-(3-((5-(4-Fluorophenyl)thiophen-2-yl)methyl)-4-methylphenyl)-tetrahydro-6-(hydroxymethyl)-2-methoxy-2H-pyran-3,4,5-triol Anti Diabetic Canagliflozin
44 1,4,8,11-Tetraazacyclotetradecane Cyclam 295-37-4
45 2-[(4-Cyanophenyl)amino]acetic acid Anti Coagulant Dabigatran 42288-26-6
46 Ethyl N-[3-amino-4-(methylamino)benzoyl]-N-pyridin-2-yl-β-alaninate Anti Coagulant Dabigatran 212322-56-0
47 ethyl 3-(2-((4-cyanophenylamino)methyl)-1-methyl-N-(pyridin-2-yl)-1H-benzo[d]imidazole-5-carboxamido)propanoate Anti Coagulant Dabigatran 211915-84-3
48 5-bromo-2-chloro-4-ethoxydiphenylmethane Anti Diabetic Dapagliflozin 461432-23-5
49 (2S,3R,4S,5S,6R)-2-(4-chloro-3-((4-ethoxybenzyl) phenyl)-6-(hydroxymethyl)-2-methoxytetrahydro-2H-pyran-3,4,5-triol Anti Diabetic Dapagliflozin
50 (S)-(-)- 2,6-diamino-4,5,6,7-tetrahydro benzothiazole Anti Parkinsonian Dex pramipexole/Pramipexole 106092-09-5
51 (R)-(+)- 2,6-diamino-4,5,6,7-tetrahydro benzothiazole Anti Parkinsonian Dex pramipexole/Pramipexole 106092-11-9
52 (±)- 2,6-diamino-4,5,6,7-tetrahydro benzothiazole Anti Parkinsonian Dex pramipexole/Pramipexole 104617-49-4
53 2-(chloromethyl)-4-methylquinazoline Anti Diabetic Linagliptin 109113-72-6
54 8-Bromo-7-(but-2-yn-1-yl)-3-methyl-3,7-dihydro-1H-purine-2,6-dione Anti Diabetic Linagliptin 666816-98-4
55 1-Bromo-2-butyne Anti Diabetic Linagliptin 3355-28-0
56 (R)-3-amino piperidine dihydrochloride Anti Diabetic Linagliptin 334618-23-4
57 8-bromo-3-methyl-1H-purine-2,6(3H,7H)-dione Anti Diabetic Linagliptin 93703-24-3
58 (S)-2-chloro-1-(2,4-dichlorophenyl)ethyl methanesulfonate Anti Fungal Luliconazole 229334-55-8
59 1-(Cyanomethyl)imidazole Anti Fungal Luliconazole 98873-55-3
60 3-(1-Piperazinyl)-1,2-benzisothiazole Anti Psychotic Lurasidone 87691-87-0
61 (1R,2R)-1,2-Cyclohexanedimethanol Anti Psychotic Lurasidone 65376-05-8
62 (3aR,4S,7R,7aS) 4,7-Methano-1H-isoindole-1,3(2H)-dione Anti Psychotic Lurasidone 14805-29-9
63 ( R)-N-(4-Nitrophenethyl)-2-hydroxy-2-phenyl acetamide Anti Muscarinic Mirabegron 521284-19-5
64 ( R)-2-(4-Nitrophenethylamino)-1-phenylethanol hydrochloride Anti Muscarinic Mirabegron
65 5-(Pyridin-2-yl)pyridin-2(1H)-one Anti Epileptic Perampanel
66 1-Phenyl-5-(pyridin-2-yl)pyridin-2(1H)-one Anti Epileptic Perampanel
67 3-Bromo-1-phenyl-5-(pyridin-2-yl)pyridin-2(1H)-one Anti Epileptic Perampanel
68 5′-(2-Cyanophenyl)-1′-phenyl-2,3′-bipyridinyl-6′(1’H)-one Anti Epileptic Perampanel 380917-97-5
69 2,4-Diamino-6-(bromomethyl)pteridine Hydrobromide Anti Cancer PralatrexateMethotrexate 73978-41-3
70 Methyl 4-(1-(methoxycarbonyl)but-3-ynyl)benzoate Anti Cancer Pralatrexate 146464-90-6
71 Methyl 4-(2-(methoxycarbonyl)-1-(2,4-diaminopteridin-6-yl)pent-4-yn-2-yl)benzoate Anti Cancer Pralatrexate 146464-91-7
72 Benzoic acid, 4-[1-[2,4-diamnio-6-pteridinyl)methyl]-3-butyn-1-yl Anti Cancer Pralatrexate 146464-93-9
73 1-[[(2R, 3S)-2-(2, 4-difluorophenyl)-3- Methyloxiranyl] methyl]-1H-1, 2, 4-triazole Anti Fungal Rauvaconazole 127000-90-2
74 Boc-3-Hydroxy-1-adamantyl-D-glycine Anti Diabetic Saxagliptin 361442-00-4
75 (1S,3S,5S)-3-(Aminocarbonyl)-2-azabicyclo[3.1.0]hexane-2-carboxylic acid tert-butyl ester Anti Diabetic Saxagliptin 361440-67-7
76 Cis-N-benzyl-3-methyl amino-4-methyl piperidine- Bis hydrochloride Rheumatoid Arthritis Tofacitinib/Tasocitinib
77 4-Chloro-7-tosyl-7H-pyrrolo[2,3,-d]pyrimidine Rheumatoid Arthritis Tofacitinib/Tasocitinib 479633-63-1
78 N-Methyl-N-((3R,4R)-4-methylpiperidin-3yl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine Rheumatoid Arthritis Tofacitinib/Tasocitinib 477600-74-1
79 4,6-dichloro-5-nitro-2-(propylthio)pyrimidine Anti Thrombotic Ticagrelor 145783-14-8
80 (1R,2S)-2-(3,4-difluorophenyl)cyclopropanamine Anti Thrombotic Ticagrelor 220352-38-5
81 2-{[(3aR,4S, 6R, 6aS)-6-amino-2, 2-dimethyltetrahydro-3aH-cyclopenta[d][1,3]-dioxol-4-yl]oxy}-1-ethol Anti Thrombotic Ticagrelor 274693-55-9
82 5-(1-Piperazinyl)-1-benzofuran-2-carboxamidehydrochloride Anti Depressant Vilazodone 183288-46-2
83 3-(4-Chlorobutyl)-1H-indole-5-carbonitrile Anti Depressant Vilazodone 143612-79-7
84 2-Chloro-1-(2-chlorophenyl)ethyl methanosulfonate Anti Fungal Lanoconazole
85 4-[(4’-Dimethyl amino)-1-(4”-fluorophenyl)-1-hydroxy butyl]-3-(hydroxy methyl) benzonitrile Antidepressant Citalopram / Escitalopram  103146-25-4
86 4-[(4’-Dimethyl amino)-1-(4”-fluorophenyl)-1-hydroxy butyl]-3-(hydroxy methyl) benzonitrile HBr Antidepressant Citalopram / Escitalopram  103146-26-5
87 4-[(4’-Dimethyl amino)-1-(4”-fluorophenyl)-1-hydroxy butyl]-3-(hydroxy methyl) benzonitrile HCl Antidepressant Citalopram / Escitalopram  717133-25-0
88 4[(4’-Dimethyl amino)-1-(4”-fluorophenyl)-1hydroxy butyl]-3-(hydroxy methyl)benzonitrile Oxalate Antidepressant Citalopram / Escitalopram 717133-32-9
89 1-[3-(dimethylamino)propyl]-1-(4-fluorophenyl)1,3-dihydroisobenzofuran-5-carbonitrile Antidepressant Citalopram / Escitalopram 59729-33-8
90 1-[3-(Dimethylamino)-propyl]-1-(4-fluoro phenyl)-5-phthalan carbonitrile HCl Antidepressant Citalopram / Escitalopram 85118-27-0
91 1-(4’-Fluoro phenyl)-1,3-dihydro iso benzofuran-5-carbonitrile Antidepressant Citalopram / Escitalopram 64169-67-1
92 5-Bromo-1-(3-dimethyl amino propyl) –1-(4’fluoro phenyl)-1,3-dihydro isobenzofuran oxalate Antidepressant Citalopram / Escitalopram
93 1-(4-bromo-2-(hydroxymethyl)phenyl)-4-(dimethylamino)-1-(4-fluorophenyl) butan-1-ol oxalate Antidepressant Citalopram / Escitalopram
94  (+)-Dipara tolouyl–d-tartaric acid salt of 4-[(4’-Dimethyl amino)-1-(4”-fluorophenyl)-1-hydroxy butyl]-3-(hydroxy methyl) benzonitrile Antidepressant Citalopram / Escitalopram 128173-53-5
95 3-N,N’-(dimethylamino)propyl chloride Hydrochloride Antidepressant Citalopram / Escitalopram 1281001
96 1,2,3,9-tetrahydro-4H-carbazol-4-one Antiemetic Ondansetron hydrochloride dihydrate 15128-52-6
97 3-Dimethyl amino-1-(2-thienyl)-1-propanone hydrochloride Antidepressant Duloxetine 5424-47-5
98 RS-N,N-Dimethyl-3-hydroxy-3-(2-thienyl)-1-propanamine Antidepressant Duloxetine 13636-02-7
99 S(-)-N,N-Dimethyl-3-hydroxy-3-(2-thienyl)-1-propanamine Antidepressant Duloxetine 132335-44-5
100 RS-N,N- Dimethyl-3-(1-Naphthalenyloxy)-3-(2-thienyl)-1-propanamine oxalate Antidepressant Duloxetine 116817-12-0
101 S-(+)-N,N-Dimethyl-3-(1-Naphthalenyloxy)-3-(2-thienyl)-1-propanamine oxalate Antidepressant Duloxetine 132335-47-8
102 (N,N-dimethyl-3-(naphthalen-1-yloxy)-3-(thiophen-2-yl)propan-1-amine Fumarate. Antidepressant Duloxetine
103 N-Methyl-3-(naphthalen-1-yloxy)-3-(thiophen-2-yl)propan-1-amine Oxalate (Racemic Duloxetine Oxalate). Antidepressant Duloxetine
104 N-(2,6-dimethylphenyl)-2-(piperazin-1-yl)acetamide Antianginals Ranolazine 5294-61-1
105 2-((2-methoxyphenoxy)methyl)oxirane Antianginals Ranolazine 2210-74-4
106 α-(meta hydroxy phenyl) ethyldimethyl amine Central Nervous System Agent Rivastigmine 105601-04-5/HCl- 5441-61-2
107 S (+)-α meta hydroxy phenyl)ethyl dimethyl amine Central Nervous System Agent Rivastigmine 139306-10-8
108 Racemic Rivastigmine hydrochloride Central Nervous System Agent Rivastigmine 105601-14-7
109 3-(1-aminoethyl)phenol Central Nervous System Agent Rivastigmine 63720-38-7
110 (S)- 3-(1-aminoethyl)phenol Central Nervous System Agent Rivastigmine 123982-81-0
111 L-Valine methyl ester hydrochloride Cardiovascular Agent Valsartan 6306-52-1
112 L-Valine benzyl ester hydrochloride Cardiovascular Agent Valsartan 2462–34-2
113 L-Valine benzyl ester p-toluene sulfonate Cardiovascular Agent Valsartan 16652-76-9
114 N-[(2′-Cyanobiphenyl-4-methyl)-(L)-Valine  methyl ester Hydrochloride Cardiovascular Agent Valsartan 482577-59-3
115 2-chloro-N-(2,6-dimethylphenyl)acetamide Anesthetic Lidiocaine 1131-01-7
116 2,2-Diphenyl-2-((R)-pyrrolidin-3-yl)acetonitrile hydrobromide Urinary Antispasmodic Darifenacin 194602-27-2
117 3-(S)-(+)-(1-carbamoyl-1,1-diphenylmethyl) pyrrolidine – L-(+)-tartrate Urinary Antispasmodic Darifenacin 134002-26-9
118 5-(2-chloroethyl)-2,3-dihydrobenzofuran Urinary Antispasmodic Darifenacin 943034-50-2
119 5-(2-bromoethyl)-2,3-dihydrobenzofuran Urinary Antispasmodic Darifenacin 127264-14-6
120 (S)-1-(2-chloroacetyl)pyrrolidine-2-carbonitrile Antidiabetics Vildagliptin 207557-35-5
122 (S)-3-Methyl-1-(2-piperidin-1-ylphenyl)butylamine Hypoglycemic Repaglinide 147769-93-5
123 (S)-Repaglinide Ethyl Ester Hypoglycemic Repaglinide 147770-06-7
124 3-(trifluoromethyl)-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyrazine hydrochloride Hypoglycemic Sitagliptin 762240-92-6
125 1-(3-(trifluoromethyl)-5,6-dihydro-[1,2,4]triazolo[4,3-a]pyrazin-7(8H)-yl)-4-(2,4,5-trifluorophenyl)butane-1,3-dione /(2Z)-4-Oxo-4-[3-(trifluoromethyl)-5,6-dihydro-[1,2,4]triazolo[4,3-a]pyrazine-7(8H)-yl]-1-(2,4,5-trifluorophenyl)butan-2-one Hypoglycemic Sitagliptin 764667-65-4
126 3,4-Dihydro-6-methyl-4-phenylchromen-2-one Urinary tract antispasmodic Tolterodine Tartrate 40546-94-9
127 3-(2-Methoxy-5-methylphenyl)-3-phenylpropan-1-ol Urinary tract antispasmodic Tolterodine Tartrate 124937-73-1
128 2-(3-(diisopropylamino)-1-phenylpropyl)-4-methylphenol (Racemic Tolterodine) 124936-74-9) Urinary tract antispasmodic Tolterodine Tartrate 124936-74-9
129 3,4-dihydro-5-hydroxyquinolin-2(1H)-one Antiglaucoma. Carteolol 30389-33-4
130 5-((oxiran-2-yl)methoxy)-3,4-dihydroquinolin-2(1H)-one Antiglaucoma. Carteolol 51781-14-7
131 3-Chloro-1-phenylpropan-1-ol Dapoxetine 100306-33-0
132 Racemic Dapoxetine Oxalate Dapoxetine
133 Racemic Dapoxetine Hydrochloride Dapoxetine 1071929-03-7
134 Dapoxetine Base Dapoxetine 119356-77-3
135 6-Chloroindolin-2-one Antipsychotic Ziprasidone 56341-37-8
136 6-Chloro-5-(2-chloroethyl)indolin-2-one Antipsychotic Ziprasidone 118289-55-7
137 Boc-D-Serine  Anticonvulsant Lacosamide 6368-20-3
138 Boc-O-Methyl-D-serine  Anticonvulsant Lacosamide 86123-95-7
139 (R)-tert-Butyl 1-(benzylamino)-3-methoxy-1-oxopropan-2-ylcarbamate  Anticonvulsant Lacosamide 880468-89-3
140 (R)-2-amino-N-benzyl-3-methoxypropanamide  Anticonvulsant Lacosamide 196601-69-1
141 N-Cbz-D-Serine  Anticonvulsant Lacosamide 6081-61-4
142 (R)-N-benzyl-2-(benzyloxycarbonylamino)-3-hydroxypropionamide  Anticonvulsant Lacosamide 219835-31-1
143  (S)- 6-Fluoro-3,4-dihydro-2H-1-benzopyran-2-carboxylic acid Antihypertensive Nebivolol 129101-36-6
144 (R )-6-Fluoro-3,4-dihydro-2H-1-benzopyran-2-carboxylic acid Antihypertensive Nebivolol 129101-37-7
145 (6-fluoro-3,4-dihydro-2H-1-benzopyran-2-yl)(piperidin-1-yl)methanone Antihypertensive Nebivolol 878208-57-2
146 6-Fluoro-3,4-dihydro-2-oxiranyl-2H-1-benzopyran (Mixture of Two Diastereomers) Antihypertensive Nebivolol 99199-90-3
147 2-(benzylamino)-1-(6-fluorochroman-2-yl)ethanol Antihypertensive Nebivolol
148 N-Benzyl Nebivolol Hydrochloride Antihypertensive Nebivolol
149 1,3-Cyclohexanedione Cardiovascular Agent Carvedilol 504-02-9
150 4-Hydroxycarbazole Cardiovascular Agent Carvedilol 52602-39-8
151 4-(2,3-Epoxypropoxy)carbazole Cardiovascular Agent Carvedilol 51997-51-4
152 2-(2-Methoxyphenoxy)ethylamine Cardiovascular Agent Carvedilol 1836-62-0
153 2-(2-Methoxyphenoxy)ethylamine HCl Cardiovascular Agent Carvedilol 64464-07-9
154 N-(2-(2-Methoxyphenoxy)ethyl)benzylamine Cardiovascular Agent Carvedilol 3246-03-5
155 N-(2-(2-Methoxyphenoxy)ethyl)benzylamine HCI Cardiovascular Agent Carvedilol 120606-08-8
156 2-[2-(2-methoxyphenoxy)ethyl]-1H-isoindole-1,3(2H)-dione Cardiovascular Agent Carvedilol 26646-63-9
157 4-[(4’-Dimethyl amino)-1-(4”-fluorophenyl)-1-hydroxy butyl]-3-(hydroxy methyl) benzonitrile Antidepressant Citalopram / Escitalopram Oxalate Diol 103146-25-4
158 4-[(4’-Dimethyl amino)-1-(4”-fluorophenyl)-1-hydroxy butyl]-3-(hydroxy methyl) benzonitrile HBr Antidepressant Citalopram / Escitalopram 103146-26-5
159 4-[(4’-Dimethyl amino)-1-(4”-fluorophenyl)-1-hydroxy butyl]-3-(hydroxy methyl) benzonitrile HCl Antidepressant Citalopram / Escitalopram 717133-25-0
160 5-Bromo-1-(3-dimethyl amino propyl) –1-(4’fluoro phenyl)-1,3-dihydro isobenzofuran oxalate Antidepressant Citalopram / Escitalopram
161 1-(4-bromo-2-(hydroxymethyl)phenyl)-4-(dimethylamino)-1-(4-fluorophenyl) butan-1-ol oxalate Antidepressant Citalopram / Escitalopram
162 3-N,N’-(dimethylamino)propyl chloride Hydrochloride Antidepressant Citalopram / Escitalopram 5407-04-5
163 (N,N-dimethyl-3-(naphthalen-1-yloxy)-3-(thiophen-2-yl)propan-1-amine Fumarate Antidepressant Duloxetine
164 N-Methyl-3-(naphthalen-1-yloxy)-3-(thiophen-2-yl)propan-1-amine Oxalate Antidepressant Racemic Duloxetine Oxalate
165 α-(meta hydroxy phenyl) ethyldimethyl amine  Central Nervous System Agent Rivastigmine 105601-04-5
166 α-(meta hydroxy phenyl) ethyldimethyl amine HCI  Central Nervous System Agent Rivastigmine 5441-61-2
167 Racemic Dapoxetine Oxalate Dapoxetine Hydrochloride
168 Diethyl-2-benzylmalonate antidiarrheal Racecadotril 607-81-8
169 Dimethyl-2-benzylmalonate antidiarrheal Racecadotril 6626-84-2
170 2-Benzylacrylic acid antidiarrheal Racecadotril 5669-19-2
171 (RS)- 6-Fluoro-3,4-dihydro-2H-1-benzopyran-2-carboxylic acid Antihypertensive Nebivolol
172 2-(benzylamino)-1-(6-fluorochroman-2-yl)ethanol Antihypertensive Nebivolol
173 N-Benzyl Nebivolol Hydrochloride Antihypertensive Nebivolol
174 N-Methyl-1-Naphthyl methyl amine hydrochloride 65473-13-4
175 N-Boc-Prolinamide 35150-07-3
176 L-Prolinamide 7531-52-4
177 N-Boc-L-Proline 15761-39-4
178 2-Methyl cyclohexane 1,3-dione 1193-55-1
179 L-Valinamide HCl 3014-80-0
180 Diethyl-D-tartrate 13811-71-7
181 L-Alanine methyl ester HCl 2491-20-5
182 L-Proline methyl ester HCl 2133-40-6
183 (S)-3-Chloroalanine methyl ester hydrochloride 112346-82-4
184 (S)-Pyrrolidine-2-carbonitrile hydrochloride 65732-69-6
185 D-Serine methyl ester hydrochloride 5874-57-7
186 N-Boc-D-serine methyl ester 95715-85-8
187 1(2-(2-chlorophenyl)acetaldehyde 4251-63-2
188 N-Boc-(S)-(-)-2-amino-1-butanol 150736-72-4
189 N-Boc-L-Valine 13734-41-3
190 N-Cbz-L-Proline 1148-11-4
191 N-Cbz-L-Valine 1149-26-4
192 (+)-O,O’-Dibenzoyl-D-tartaric acid monohydrate 80822-15-7
193 (+)-O,O’-Dibenzoyl-D-tartaric acid monohydrate anhydrous 17026-42-5
194 (-)-O,O’-Dibenzoyl-L-tartaric acid monohydrate 62708-56-9
195 (-)-O,O’-Dibenzoyl-L-tartaric acid monohydrate anhydrous 2743-38-6
196 (-)-O,O’-Di-p-toluoyl-L-Tartaric acid Monohydrate 71607-31-3
197 (-)-O,O’-Di-p-toluoyl-L-Tartaric acid Monohydrate anhydrous 32634-66-5
198 (+)-O,O’-Di-p-toluoyl-D-Tartaric acid Monohydrate 71607-32-4
199 (+)-O,O’-Di-p-toluoyl-D-Tartaric acid Monohydrate anhydrous 32634-68-7
200 S-(-)-2-(3,4-Dimthoxybenzyl)-2-hydrazinyl propionic acid  ( Dimethoxy carbidopa)
201 S-(+)-2-Phenyl propionic acid 7782-24-3
202 9-Phenylcarbazole 1150-62-5
203 ortho-Phthalaldehyde 643-79-8
204 3,6-Dibromo-9-Phenylcarbazole 57103-20-5
205 (S) – (+) – 2 – Cholorophenyn glycine methyl ester Antiplatelet drug Clopidogrel Bisulphate 141109-14-0
206 (+) – Methyl-α-(2-thienylethamino)(2-chlorophenyl) acetate hydrochloride Antiplatelet drug Clopidogrel Bisulphate 141109-19-5
207 4,5,6,7 – Tetrahydrothieno [3,2,c] pyridine hydrochloride Antiplatelet drug Clopidogrel Bisulphate 28783-41-7
208 3- (Trifluoromethyl)-5,6, 7,8- tetrahydro [1, 2, 4] triazolo [4, 3-a] Pyrazine hydrochloride( 1 -4) Hypoglycemic Sitagliptin 486460-21-3
209 (3R)T-BUTOXYCARBONY AMINO -4-(2,4,5- TRIFLUOROPHENYL) BUTANOIC ACID Hypoglycemic Sitagliptin 486460-00-8
210 (2Z)-4-Oxo-4-[3-(trifluoromethyl)-5,6-dihydro-[1,2,4]triazolo[4,3-a]pyrazine-7(8H-yl]-1-(2,4,5-trifluorophenyl)but-2-en-2-amine Hypoglycemic Sitagliptin 767340-03-4
211 4-Hydrazino-N-methylbenzene methane sulphonamide Vascular headache suppressant Sumatriptan 88933-16-8
212 4-Chloro 1-hydroxybutane sulphonic acid Vascular headache suppressant Sumatriptan 54322-20-2
213 1-(4-Hydrazinophenyl) methyl-1,2,4-triazole Dihydrochloride  Antimigraine Rizatriptan 212248-62-9
214 4-N,N-Dimethyl amino butanal dimethyl acetal  Antimigraine Rizatriptan 19718-92-4
215 4-(4-Aminophenyl) MORPHOLIN-3-one Anticoagulant. Rivaroxaban 438056-69-0
216 5-Chlorothiophene-2-carboxylic acid Anticoagulant. Rivaroxaban 24065-33-6
217 Ethyl 3- (pyridin-2- ylamino) propanoate Anticoagulant. Dabigatran 103041-38-9
218 3-HYDROXY-I-AMINOADAMANTANE  Antidiabetics. Vildagliptin 702-82-9
219 3-Fluoro-4-morpholinyl aniline  Antibiotic Linezolid 93246-53-8
220 4-(Chloromethyl)-2,2-dimethyl-1,3-dioxolane  Antibiotic Linezolid 4362-40-7
221 2-MERCAPTO-5-METHOXY BENZIMIDAZOLE (Omeprazole-Benzimidazole) Omeprazole 37052-78-1
222 2-CHLORO-METHYL-3,5-DIMETHYL-4-METHOXY PYRIDINE HCL (Omeprazole Chloro Compound) Omeprazole 86604-75-3
223 5-METHOXY-2-[[(3,5-DIMETHYL-4-METHOXY-2-PYRIDINYL)METHL]THIO]-1H BENZIMIDAZOLE (omeprazole sulphide) Omeprazole 73590-85-9
224 2-HYDROXY METHYL-3,5-DIMETHYL-4-METHOXY PYRIDINE (Omeprazole Intermediate) Omeprazole 86604-78-6
225 2-CHLOROMETHYL 3,4-DIMETHOXY PYRIDINE HYDROCHLORIDE(Pantoprazole Chloro Compound) Gastric Acid Secretion Inhibitor Pantoprazole 72830-09-2
226 5-DIFLOURO METHOXY[[[3,4-DIMETHOXY-2-PYRIDINYL]METHYL]THIO]-1H-BEZIMIDAZOLE(pantoprazole sulphide) Gastric Acid Secretion Inhibitor Pantoprazole 102625-64-9
227 2-MERCAPTO-5-DIFLOURO METHOXY BENZIMIDAZOLE (Pantoprazole Benzimidazole) Gastric Acid Secretion Inhibitor Pantoprazole 97963-62-7
228 L(+)- Di Ethyl Tartarate 87-91-2
229 2-CHLORO METHYL-4-(3-METHOXY PROPOXY)-3-METHYL PYRIDINE HYDROCHLORIDE(Rabeprazole Chloro compound) Gastric Acid Secretion Inhibitor Rabeprazole 153259-31-5
230 2-[[[3-METHYL-4-(3-METHOXYPROPOXY)-2-PYRIDYL]METHYL]THIO]-1H-BENZIMIDAZOLE; 2-{[4-(3-METHOXYPROPOXY)-3-METHYLPYRIDINE-2-YL]-METHYTHIO}-1H-BENZIMIDAZOLE (Rabeprazole Sulphide) Gastric Acid Secretion Inhibitor Rabeprazole 117977-21-6
231 Ammonium Sulphate 7783-20-2
232 TRISODIUM ORTHOPHOSPHATE (TSP) 96337-98-3
233 SODIUM NITRITE 7632-00-0
234 DISODIUM ORTHO PHOSPHATE 7632-05-5
235 DI AMMONIUM PHOSPHATE 7783-28-0
236 2(2,4 Difluorophenyl)-1-(4-amino)-1H-1,2,4-triazole-1-yl)-ethanone Hydrochloride Antifungal Fluconazole
237 1-(2,4-Difluorophenyl)-1-(1H-1,2,4-triazole-1yl)-ethanone(DFTA) Antifungal Fluconazole
Voriconazole
86404-63-9
238 2-(2,4-Difluorophenyl)-1-(1H-1,2,4-triazole-1yl)2,3Epoxy propane-Methane sulphonate (EPOXY MESYLATE) Antifungal Fluconazole 86386-77-8
239 6,6-Dimethylhept-1-en-4-yn-3-ol Antifungal Terbinafine 78629-20-6
240 1-Chloro-6,6-dimethylhept-2-en-4-yne Antifungal Terbinafine 83554-69-2
241 N-(1-naphthyl methyl)methylamine (Free Base) Antifungal Terbinafine 14489-75-9
242 (2E) N,6,6_Trimethyl-N-(naphthalene-1-ylmethyl)Hept-2-en-4-yn-1-amine Antifungal Terbinafine 91161-71-6
243 2-n-butyl-4-chloro-1[(2’cyanobiphenyl-4-yl)methyl]-5-hydroxymethyl-imidazole Cardiovascular Agent Losartan Potassium 114772-55-3
244 2-butyl-4-chloro-1-[[2′-(1 H-tetrazole-5-yl)(1,1′-biphenyl)-4yl]methyl]-1HImidazole-5-methanol(Losartan) Cardiovascular Agent Losartan Potassium 114798-26-4
245 2-n-Butyl-4-chloro-5-hydroxy methyl-1-[2′-[(2-triphenylmethyl) tetrazole-5-yl] biphenyl-4-yl]methyl imidazole (Trityl Losartan) Cardiovascular Agent Losartan Potassium 133909-99-6
246 4-(1H-1,2,4-Triazol-1-yl methyl) Benzeneamine Antimigraine Rizatriptan
247 4-(1H-1,2,4-Triazol-1-yl methyl) phenyl hydrazine dihydrochloride Antimigraine Rizatriptan 154748-67-1
248 2-(n-Butyl)-3-[2′-(cyano)biphenyl-4-yl]methyl-1,3-diazaspiro[4,4]non-1-en-4-one Cardiovascular Agent Irbesartan 138401-24-8
249 2-Butyl-3-[2′-triphenylmethyltetrazol-5-yl)-biphenyl-4-yl methyl]-1,3-diazaspiro[4,4] non-1-ene-4-one (Trityl Irbesartan) Cardiovascular Agent Irbesartan 138402-10-5
250 N,N-Dimethyl-1-phenyl-3-(1-napthalenyloxy)propanamine oxalic acid salt (Racemic Dapoxetine oxalate) Dapoxetine
251 [2-(2-Phthalimido ethoxy methyl-3-Carbo ethoxy-1-(chlorophenyl)-5-carbomethoxy-6-methyl-1,4-dihydro pyridine(phthaloyl Amlodipine)  Antihypertensive Amolidipine Besylate 88150-62-3
252 Amlodipine Base  Antihypertensive Amolidipine Besylate 88150-47-4
253 N-(triphenyl methyl)-5-(4′-bromo methyl bi phenyl 2-yl)tetrazole [TTBB] Cardiovascular Agent Olmesartan 133051-88-4
254 (5-Methyl-2-Oxo-1,3-Dioxolen-4-yl)-Methyl-4-(1-hydroxy-1-Methyl-ethyl)-2-propyl-1-[4-[2-trityltrizole-5-yl)-Phenyl]-phenyl]-Methylimidazole-5-Carboxylate[trityl olmesartan medoxomil] Cardiovascular Agent Olmesartan 144690-92-6
255 3-(N-methyl-N-pentylamine)-propionic acid hydrochloride salt Calcium Regulator Ibandronate
256 2-Hydroxy methyl-4-(3-methoxy propoxy)-3-methyl-pyridine hydrochloride Gastric antisecretory agent Rabeprazole Hydroxy 118175-10-3
257 2,3,4,5-Bis-0-(1-Methyl ethylidine)-Fructopyranose-Azido sulphate (TP-II) Anticonvulsant Topiramate 106881-35-0
258 [(2R, 5R)-5-Hydroxy-[1,3]-Oxathiolane-2-Carboxylic acid, 2S-isopropyl-5R-methyl-1R-cyclohexyl ester] (ECE) Anti- Hepatitis Agents. Lamivudine 147027-10-9
259 (L)-Menthyl Glyoxylate Monohydrate (MGH) Anti- Hepatitis Agents. Lamivudine 11969-64-3
260 (L)-Menthyl Glyoxylate Monohydrate (MGH-I) Anti- Hepatitis Agents. Lamivudine 26315-61-7
261 (2R, 5R)-5-(4-Amino-5-Fluoro-2-oxo-2H-pyrimidin-1-yl)-[1,3]oxathiolane-2-carboxylic acid, 2S-Isopropyl-5R-methyl-1RCyclohexylester (FCME)  Anti-Infective Agent Emtricitabine 764659-72-5
262 3-Azido-5-O-Trityl thymidine Antiretroviral Zidovudine
263 9-(2-Phosphonyl methoxypropyl) Adenine Antiretroviral Tenofovir 147127-20-6
264 4-(1-Pyrrolidinylsulphonylmethyl)-phenylhydrazine hydrochloride Antimigraine Almotriptan Malate 334981-11-2
265 (1S,2S,3R,5S)-Pinanediol-1-ammoniumtrifluoroacetate-3-methylbutane-1-boronate Antineoplastic Agent Bortezomib 179324-87-9
266 5-Bromo-3-(((R)-1-methylpyrrolidin-2-yl)methyl)-1H-indole Antimigraine Eletriptan Hydrobromide 143322-57-0
267 1-(Vinylsulfonyl)benzene (OR) Phenyl Vinyl Sulfone Antimigraine Eletriptan Hydrobromide 5535-48-8
268 (1R,3R)-Methyl-1-(benzo[d][1,3]dioxol-5-yl)-2-(2-chloroacetyl)-2,3,4,9-tetrahydro-1H- pyrido[3,4-b]indole-3-carboxylate Erectile Dysfunction Agent Tadalafil 171489-59-1
269 (S)-4-(4-Aminobenzyl)-2-oxazolidinone Antimigraine Zolmitriptan 152305-23-2
270 (R)-N-[[3-[3-Fluoro-4-morpholinyl]phenyl]-2-oxo-5-oxazolidinyl]methanol  Antibiotic Linezolid 168828-82-8
271 4 – (3,4 -Dichloro Phenyl) -3,4-Dihydro -1(2H) – Naphthalenone / TETRALONE Antidepressant Sertraline Hcl 79836-44-5
272 N-Methyl – 4-( 3, 4 -Dichloro Phenyl) -1,2,3,4 Tetrahydro –1-  Napthalene Imine / TETRALONE – IMINE Antidepressant Sertraline Hcl 79617-89-3
273 N-Methyl-4-(3,4 –Dichloro Phenyl) -1,2,3,4Tetrahydro – 1 – Napthalene Amine/ TETRALONE AMINE Antidepressant Sertraline Hcl 140631-53-4
274 Formamidine Acetate Antifungal Itraconazole & Voriconazole 3473-63-0
275 Triphenyl Amine 603-34-9
276 4,4 – Dimethyl Triphenyl Amine 20440-95-3
277 4 CNA – 4 Chloro 1,8 Naphthaline Anhydride 4053-08-1
278 6 DDQ – 6,7 Dimethoxy 3,4 Dihydro Isoquinaline 20232-39-7
279 4 SNA – 4-Sulphono naphthalic anhydride 71501-16-1
280 Iodo Benzene 591-50-4
281 4-IodoToluene 624-31-7
282 Closantel Amine 61437-85-2
283 Alpha Tetralone 529-34-0
284 (1S,3S)-(3-Aminocyclopentyl) methanol Antiretroviral agent Abacavir Sulfate 664341-71-3
285 N-(2-Amino-4,6-dichloro-5-pyrimidinyl) formamide Antiretroviral agent Abacavir Sulfate 171887-03-9
286 2-Azabicyclo[2.2.1]hept-5-en-3-one (Vince lactam) Antiretroviral agent Abacavir Sulfate 49805-30-3
287 3-Amino-2,2-dimethylpropanamide  Antihypertensive Aliskiren 324763-51-1
288 (S)-4-Benzyl-3-((S)2-((R-2-bromo-2((2S,4S)-4-isopropyl-5-oxo-tetrahydro-furan-2-yl)-3-methyl-butyryl)-oxaxolidin-2-one  Antihypertensive Aliskiren 173154-00-2
289 (S)-4-Benzyl-2-oxazolidinone  Antihypertensive Aliskiren 90719-32-7
290 4-Bromo-1-methoxy-2-(3-methoxypropoxy)-benzene  Antihypertensive Aliskiren 173336-76-0
291 (R)-4-(2-(Chloromethyl)-3-methylbutyl)-1-methoxy-2-(3-methoxypropoxy)benzene  Antihypertensive Aliskiren 324763-39-5
292 trans-1,4-Dibromo-2-ene  Antihypertensivee Aliskiren 821-06-7
293 3-Isovaleroyl-4-(R)-benzyl-oxazolidin-2-one  Antihypertensive Aliskiren 145589-03-3
295 tert-Butyl [(1S,2R)-1-benzyl-2-hydroxy-3-(isobutylamino)propyl]carbamate Antiviral Darunavir 160232-08-6
296 tert-Butyl [(1S,2R)-1-benzyl-2-hydroxy-3-[isobutyl[(4-nitrophenyl)sulfonyl]amino]propyl]carbamate Antiviral Darunavir 191226-98-9
297 [(1S,2R)-1-Benzyl-2-hydroxy-3-[isobutyl-[(4-aminophenyl)sulfonyl]amino]propyl]-carbamic Acid tert-Butyl Ester Antiviral Darunavir 183004-94-6
298 [(3R,3aS,6aR)-Hydroxyhexahydrofuro[2,3-β]furanyl succinimidyl carbonate Antiviral Darunavir 253265-97-3
299 4-Nitrobenzenesulfonyl chloride Antiviral Darunavir 98-74-8
300 (S)-(-)-3-(N-Methylamino)-1-(2-thienyl)-1-propanol Antidepressant Duloxetine Hydrochloride 116539-55-0
301 (1S,2S,3S,5S)-5-(2-Amino-6-(benzyloxy)-9H-purin-9-yl)-3-(benzyloxy)-2-(benzyloxymethyl)cyclopentanol Antiviral Entecavir 142217-77-4
302 2-Amino-1,9-dihydro-9-[(1S,3R,4S)-4-(benzyloxy)-3-(benzyloxymethyl)-2-methylenecyclopentyl]-6H-purin-6-one Antiviral Entecavir 142217-81-0
303 (2R,3S,5S)-3-(Benzyloxy)-5-[2-[[(4-methoxyphenyl)diphenylmethyl]amino]-6-(phenylmethoxy)-9H-purin-9-yl]-2-(benzyloxymethyl)cyclopentanol Antiviral Entecavir 142217-78-5
304 6-(Benzyloxy)-9-[(1S,3R,4S)-2-methylene-4-(phenylmethoxy)-3-[(phenylmethoxy)methyl]cyclopentyl]-9h-purine-2 amine Antiviral Entecavir 204845-95-4
305 (1S,2R,3S,5R)-3-(Phenylmethoxy)-2-[(phenylmethoxy)methyl]-6-oxabicyclo[3.1.0]hexane Antiviral Entecavir 110567-22-1
306 Ethyl 2-(3-cyano-4-isobutoxyphenyl)-4-methyl-5-thiazolecarboxylate Antigout Febuxostat 160844-75-7
307 Ethyl 2-(3-formyl-4-hydroxyphenyl)-4-methylthiazole-5-carboxylate Antigout Febuxostat 161798-01-2
308 Ethyl 2-(3-formyl-4-isobutoxyphenyl)-4-methylthiazole-5-carboxylate Antigout Febuxostat 161798-03-4
309 Benzenesulfonamide,N-[(2R,3S)-3-amino-2-hydroxy-4-phenylbutyl]-N-(2-methylpropyl)-4-nitro Antiretroviral agent Fosamprenavir 251105-80-3
310 (2R,3S)-3-(tert-Butoxycarbonyl)amino-1,2-epoxy-4-phenylbutane Antiretroviral agent Fosamprenavir 98760-08-8
311 (S)-(+)-3-Hydroxytetrahydro furan Antiretroviral agent Fosamprenavir 86087-23-2
312 [(1S,2R)-3-[[(4-Nitrophenyl)sulfonyl](2-methylpropyl)amino]-2-hydroxy-1-phenylmethyl)propyl]carbamic acid,(3S)-tetrahydro-3-furanyl ester Antiretroviral agent Fosamprenavir 160231-69-6
313 2-(2-(3(S)-(3-(2-(7-Chloro-2-quinolinyl)ethenyl)phenyl)-3-hydroxy propyl)phenyl)-2-propanol Antiasthmatic Montelukast Sodium 142569-70-8
314 1-(Mercaptomethyl)-cyclopropaneacetic acid Antiasthmatic Montelukast Sodium 162515-68-6
315 Methyl 2-[(3S)-3-[3-[(1E)-2-(7-chloro-2-quinolinyl)ethenyl]phenyl]-3-hydroxy propyl] benzoate Antiasthmatic Montelukast Sodium 181139-72-0
316 Methyl 2-(3-{(E)-3-[2-(7-chloro-2-quinolyl)vinyl]phenyl}-3-oxopropyl)benzoate Antiasthmatic Montelukast Sodium 149968-11-6
317 (+)-3-(Carbamoy methyl)-5-methylhexanoic acid Neuropathic Pain Agent Pregabalin 181289-15-6
318 R-(-)-3-Carbamoy methyl)-5-methylhexanoic acid Neuropathic Pain Agent Pregabalin 181289-33-8
319 Epichlorohydrin  Phosphate Binder. Sevelamer Hydrochloride 106-89-8
320 Poly (allylamine hydrochloride)  Phosphate Binder. Sevelamer Hydrochloride 71550-12-4
321 Sevelamer carbonate  Phosphate Binder. Sevelamer Hydrochloride 845273-93-0
322 D-Tryptophan methyl ester hydrochloride Erectile Dysfunction Agent Tadalafil 14907-27-8
323 N-Acetyl ethylene urea Skeletal Muscle Relaxant Tizanidine 5391-39-9
324 4-Amino-5-chloro-2,1,3-benzothiadiazole Skeletal Muscle Relaxant Tizanidine 115398-34-0
325 Ethylene urea Skeletal Muscle Relaxant Tizanidine 120-93-4
326 2,4,6-Trichloro-5-Nitropyrimidine 4359-87-9
327 3-Oxocyclobutane Carboxylic Acid 23761-23-1
328 Cyclooctanone 502-49-8
329 Zolpidic Acid 189005-44-5
330 S-(-)-3-TERTIARY BUTYNYL AMINO 1,2 PROPIONIC DIOL Antihypertensive, vascular headache suppressant,
antiglaucoma agent
Timolol Maleate 189005-44-5
331 3-MORPHOLINO-4-CHLORO-1,2,5-THIADIAZOLE Antihypertensive, vascular headache suppressant,
antiglaucoma agent
Timolol Maleate
332 4-Nitro ortho Phenelendiamine Antiglaucoma Brimonidine Tartrate